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RO 3280
CAS No. 1062243-51-9
RO 3280 ( RO3280; RO-3280; RO 3280; Ro5203280 )
产品货号. M10275 CAS No. 1062243-51-9
RO3280 is a potent, highly selective inhibitor of Polo-like kinase 1 (PLK1)
纯度: >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥794 | 有现货 |
|
| 5MG | ￥1183 | 有现货 |
|
| 10MG | ￥1604 | 有现货 |
|
| 25MG | ￥3491 | 有现货 |
|
| 100MG | 获取报价 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称RO 3280
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述RO3280 is a potent, highly selective inhibitor of Polo-like kinase 1 (PLK1)
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产品描述RO3280 is a potent, highly selective inhibitor of Polo-like kinase 1 (PLK1) with IC50 of 3nM.
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同义词RO3280; RO-3280; RO 3280; Ro5203280
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通路Cell Cycle/DNA Damage
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靶点PLK
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受体PLK1
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研究领域Cancer
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适应症——
化学信息
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CAS Number1062243-51-9
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分子量543.61
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分子式C27H35F2N7O3
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纯度>98%(HPLC)
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溶解度Ethanol: 100 mg/mL (183.95 mM); DMSO: 100 mg/mL (183.95 mM)
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SMILESO=C(NC1CCN(C)CC1)C2=CC=C(NC3=NC=C(N4C)C(N(C5CCCC5)CC(F)(F)C4=O)=N3)C(OC)=C2
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化学全称4-((9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Chen S, et al. Bioorg Med Chem Lett, 2012, 22(2), 1247-1250.
产品手册
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